Open access
Jul 2026
Structural and Biophysical Characterization of Aminobenzo[d]isothiazole 1,1-Dioxide SOS1 Ligands
Comparative analysis further delineates vector requirements for productive engagement of KRAS-facing regions, providing a structure-based framework for future optimization of aminobenzo[d]isothiazole 1,1-dioxide SOS1 ligands.
Thiago Moreira Pereira, Atilio Reyes Romero, M. van der Laan et al.
· ACS Medicinal Chemistry Lett... · 0 citations