5-Carboxamide-Substituted Barbituric Acids: Promising Scaffolds for Drug Development against Mycobacterium tuberculosis.
The continued spread of drug-resistant Mycobacterium tuberculosis (Mtb) necessitates the development of new chemotypes with novel modes of action. Here, we report 5-carboxamide-substituted barbituric acid as a promising scaffold for developing new drugs against Mtb. Fenoxacrim, the initial hit compound identified throu...