Review
Sep 2026
Precision covalent chemistry: Advances in selectivity-driven covalent drug design over the past five years.
Five synergistic tactics to boost covalent inhibitor selectivity are summarized, and these innovations validate kinact/Ki as a unified rule balancing efficacy and selectivity.
Shang-Jun Bai, Meng-Han Gao, Qi-Dong You et al.
· European journal of medicina... · 0 citations