Open access
Aug 2026
Molecular Striptease of a Thiadiazolopyrimidine Hit Yields a Streamlined, Artifact-Free NADPH Mimic for NOX Inhibition
Compound 5, although aqueous solubility issues limited its cellular antiproliferative performance, represents a specific, artifact-free architectural starting point for future selective NOX inhibitor development.
Emanuele Fabbrizi, Andrea Mancini, Chiara Lambona et al.
· ACS Medicinal Chemistry Lett... · 0 citations