Author

L. Petri

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Open access Sep 2026

Fragment‐Based Screening of Heterocyclic Electrophiles Identified Acrylamide Bioisoteres for Covalent KRasG12C Inhibitors

Covalent fragment approaches gained increasing attention in medicinal chemistry. Our covalent heterocyclic fragment library (Covalent MiniFrags) consisting of five and six membered heterocycles was screened against the oncogenic target KRasG12C. First, we detected the labeling of cysteine residues by Ellman's free thio...

Nikolett Péczka, Aaron B. Keeley, Péter Ábrányi-Balogh et al. · Archiv der Pharmazie · 0 citations

Review Open access Aug 2026

Disulfide rebridging platforms for site-specific ADC conjugation

Antibody–drug conjugates (ADCs) have emerged as a transformative class of targeted therapeutics, combining the exquisite specificity of monoclonal antibodies with the potency of small-molecule cytotoxic payloads. While numerous strategies exist to generate ADCs, site-specific conjugation methods have gained prominence...

L. Petri, Írisz K. Kovács, Blanka J Kiss et al. · RSC Chemical Biology · 0 citations