Synthesis, Antifungal Activity, and Plant Systemic Mobility of Amino Acid Conjugates of a Thiasporine A-Derived Phenylthiazole Scaffold
To develop fungicidal candidates with both high antifungal activity and phloem mobility, a total of 34 2-[2-(trifluoromethoxy)phenyl]thiazole-4-carbonyl amino acid and amino acid ester conjugates were designed and synthesized. Their structures were characterized by 1H NMR, 13C NMR, and HRMS. Their in vitro antifungal a...